Articolul-1

COMMUNITY DENTISTRY                                                                                                                                     www.stomaeduj.com




EFFICACY OF BIOFLAVONOIDS OF FLAVOBAC™




                                                                                                                                                      Original Articles
AGAINST SEVERE ACUTE RESPIRATORY SYNDROME -
CORONAVIRUS 2 IN VITRO
                           1a                               2b                            3c                         4d
Abdelahhad Barbour               , Lynda Gail Darlington , Michelle Mendenhall                 , Henriette Lerner          ,
                       1,5,6e*
Michael Glogauer
1
 Faculty of Dentistry, University of Toronto, Toronto, ON, Canada, M5G 1G6
2
  Department of Internal Medicine, Ashtead Hospital, Ashtead, UK
3
  Institute for Antiviral Research, Utah State University Logan, UT, USA
4
  Goethe University, Frankfurt, GER
5
  Department of Dental Oncology, Maxillofacial and Ocular Prosthetics, Princess Margaret Cancer Centre, Toronto, ON, Canada, M5G 2M9
6
  Oral Science International Montreal, Canada
a
  DaMSc, PhD, Postdoctoral Fellow; e-mail: abdelahhad.barbour@utoronto.ca; ORCIDiD: https://orcid.org/0000-0003-0184-8890.
b
   MD, FRCP, e-mail: gail.darlington1@nhs.net
c
  MSc; e-mail: michelle.mendenhall@usu.edu; ORCIDiD: https://orcid.org/0000-0001-6417-0648.
d
  DDS; e-mail: h-lerner@web.de ORCIDiD: https://orcid.org/0000-0002-4894-9560
e
  DDS, PhD, Professor; e-mail: michael.glogauer@utoronto.ca; ORCIDiD: https://orcid.org/0000-0002-6248-5977
ABSTRACT                                                                          https://doi.org/10.25241/stomaeduj.2021.8(2).art.1
Introduction The Severe Acute Respiratory Syndrome-Coronavirus 2 (SARS-CoV-2) is responsible for the
global pandemic of Coronavirus disease-2019 (COVID-19). Human-to-human transmission occurs mainly
through the aerosolization of respiratory droplets. Improved antisepsis of human and non-human surfaces
has been identified as a key feature of transmission reduction. Flavobac, a complex of soluble bioflavonoids
and hydroxylated phenolic structures used in oral care products, has demonstrated efficacy to act against
microorganisms. This study evaluated nasal and oral antiseptic formulations of FLAVOBAC for the virucidal
activity against SARS-CoV-2.
Methodology FLAVOBAC nasal antiseptic formulations and FLAVOBAC oral rinse antiseptic formulations
from 1-10% concentrations were assayed for virucidal efficacy against the SARS-CoV-2 virus. SARS-CoV-2 was
exposed directly to the test compound for 60 seconds or 5 minutes. Compounds were then neutralized, and
the surviving virus was quantified.
Results All concentrations of nasal antiseptics and oral rinse antiseptics evaluated completely inactivated
the SARS-CoV-2 virus.
Conclusion Nasal and oral FLAVOBAC solutions are effective at inactivating the SARS-CoV-2 virus at a variety
of concentrations after 60-second or 5-minute exposure times. The formulations tested have the potential to
reduce the transmission of SARS-CoV-2 if used for nasal/oral decontamination, or surface decontamination
in known or suspected cases of COVID-19.
KEYWORDS
Bioflavonoid; COVID-19; Flavobac, SARS-COV-2; Virucidal Activity.
1. INTRODUCTION                                                                swabs) are highest at the time of, soon after, or
                                                                               before symptoms and SARS-CoV-2 RNA are detected
The emergence of the novel human Severe Acute                                  in saliva and throat swab specimens in recovered
                                                                               patients 5 to >40 days following hospital discharge
Respiratory Syndrome CoronaVirus-2 (SARS-Cov-2)
                                                                               [6]. Furthermore, live SARS-CoV-2 was isolated from
has caused drastic damage to the globe with a
                                                                               throat swab specimens, indicating viral replication
dramatic loss of human life worldwide. To date
                                                                               and shedding are active in tissues of the upper
(4 June 2021), approximately 172 million cases                                 respiratory tract where SARS-CoV-2 is not thought
have been confirmed with over 3.7 million deaths                               to replicate [7]. SARS-CoV-2 appears to remain
according to WHO [1]. Previous studies confirmed                               viable while suspended in aerosols for ~3h and on
that viral loads are high in the nasal cavity,                                 surfaces for days possibly indicating disease spread
nasopharynx, and oropharynx [2-5]. SARS-CoV-2                                  might occur even at considerable distances and in
viral RNA levels (measured in saliva, throat and nasal                         enclosed spaces with poor ventilation [8].
                OPEN ACCESS This is an Open Access article under the CC BY-NC 4.0 license.
                Peer-Reviewed Article
    Citation: Barbour A, Darlington LG, Mendenhall M, Lerner H, Glogauer M. Efficacy of Bioflavonoids of FLAVOBAC™ Against Severe Acute Respiratory
    Syndrome-Coronavirus 2 In Vitro. Stoma Edu J. 2021;8(2):95-99
    Received: May 11, 2021; Revised: OJune 03, 2021 Accepted: June 08, 2021 Published: June 10, 2021
    *Corresponding author: Prof. Dr. Michael Glogauer, DDS, PhD
    Department of Dental Oncology, Maxillofacial and Ocular Prosthetics, Princess Margaret Cancer Centre, Toronto, ON, Canada, M5G 2M9
    Tel. Fax: (905)973-0664; XYZ; e-mail: michael.glogauer@utoronto.ca




Stoma Edu J. 2021;8(2): 95-99                                                                      pISSN 2360-2406; eISSN 2502-0285                      95
                    Efficacy of FLAVOBAC™ against SARS-CoV-2
www.stomaeduj.com



                    Furthermore, among genetically related coronaviru-                             virucidal activity of commercially available 2-5%
Original Articles
                    ses, SARS-CoV-2 is predicted to have the hardest                               Flavobac solutions against the human novel SARS-
                    protective outer shell against degradative enzymes                             CoV-2 strain SARS-CoV-2, USA-WA1/2020. We report
                    thus contributing to its high resilience in saliva,                            here the first anti-SARS-CoV-2 evaluation of a na-
                    other body fluids, and outside the body [9]. Despite                           sal and oral rinse antiseptic containing Flavobac
                    many clinical trials that have been conducted for                              which has been developed specifically for routine
                    the treatment of COVID-19, no antiviral has been                               intranasal or oral use.
                    verified to be effective for COVID-19. Conventional
                    antiviral drugs including ribavirin and favipiravir and                        2. METHODS
                    other anti-inflammatory agents are currently used
                    in clinical settings against the severe cases of SARS-
                                                                                                   2.1. Virus culture and biosafety and test compounds
                    CoV-2 infections [10]. On the other hand, increased
                    interests in plant-based natural products belonging                            SARS-CoV-2, USA-WA1/2020 strain obtained from
                    to the flavonoids class have emerged as an attractive                          the World Reference Center for Emerging Viruses
                    option of treatment. The low cytotoxicity and                                  and Arboviruses (WRCEVA), was used in this study
                    synergy with other effective drugs make flavonoids                             for the virucidal activity of Flavobac. The virus
                    an ideal candidate to interfere with the life cycle of                         stock was prepared by passaging three times in
                    the virus. Several flavonoids have been shown to                               Vero 76 (ATCC, CRL-1587) cells. The media was
                    exhibit significant antiviral properties in in vitro and                       MEM supplemented with 2% fetal bovine serum
                    in vivo studies [11-13]. Bioflavonoids are naturally                           (FBS, Cytvia) and 50 μg/mL gentamicin (Sigma).
                    present in plants, fruit and vegetables, there are over                        Viral cultures were carried out in a biosafety level
                    6000 identified having a wide range of uses including                          3 (BSL-3) following standard operating procedures
                    antioxidants & food ingredients. Flavonoids com-                               approved by the USU Biohazards Committee,
                    prise a group of naturally occurring compounds                                 Institute for Antiviral Research, Utah State University,
                    that are among the most ubiquitous in the plant                                USA. Nasal antiseptic solutions and oral rinse
                    kingdom [14]. They are found in every family and                               antiseptic solutions consisting of aqueous Flavobac
                    nearly every species of the higher plants and they                             BCL concentrate as the sole active ingredient and
                    have extensive biological properties that promote                              OSI-20210203 oropharyngeal spray solution
                    human health and help reduce the risk of diseases.                             consisting of aqueous Flavobac 2% (A) and 5% (B)
                    Bioflavonoids have demonstrated their capacity to                              and other natural ingredients were supplied by Oral
                    act against bacteria, fungi, and viruses [12,15,16].                           Science International (Montreal, Canada).
                    Flavobac (Trademark of Citrox Bioscience Ltd) is a
                    natural product extracted from bitter oranges and
                                                                                                   2.2. Virucidal Assay
                    composed of soluble bioflavonoids and hydroxylated
                    phenolic structures. Flavobac is developed as nasal                            Flavobac BCL concentrate was diluted to 10%, 5%,
                    and oral rinse antiseptic formulations and besides                             2%, or 1% in the test media and OSI-20210203
                    its potent antibacterial activity against a tandem                             samples were tested at full strength. Prepared test
                    array of bacterial pathogens [15], it showed to have                           compounds were mixed with the virus stock solution
                    a strong virucidal efficacy against many viruses in                            (approximately 5.5 log10 CCID50 per 0.1 mL) at a
                    vitro (unpublished data).                                                      volume ratio of 9:1 (v/v). Each concentration was
                    In the current study, we hypothesized that                                     tested in triplicate. The Test media was added to
                    bioflavonoids as active ingredients in the Flavobac                            one tube of each prepared concentration to serve
                    may have virucidal activities against SARS-CoV-2                               as toxicity controls. Water was tested in parallel as a
                    which may enable a new application for protection                              negative control. The prepared test compound and
                    against COVID-19. We report for the first time the                             the virus solution mixtures were incubated at room
                        Table 1. Virucidal efficacy against SARS-CoV-2 after contact with the virus at 22 ± 2°C.

                        Compound                             Contact Time          Cytotoxcicity1           Neut.       Virus            Virus               LRV4
                                                                                                            Ctrl.2      Titer3           Titer3
                        FLAVOBAC BCL 10%                     1 min                 1/100                 None        <2.7             4.6             >1.9

                        FLAVOBAC BCL 5%                      1 min                 1/100                 None        <2.7             4.6             >1.9
                        FLAVOBAC BCL 2%                      1 min                 1/10n                 None        <1.7             14.6            >2.9
                        FLAVOBAC BCL 1%                      1 min                 1/10                  None        <1.7             4.6             >2.9
                        OSI-20210203A                        5 min                 1/10                  None        <1.7             4.7             > 3.0
                        OSI-20210203B                        5 min                 1/10                  None        <1.7             4.7             > 3.0
                    1
                      Cytotoxicity indicates the highest dilution of the endpoint titer where full (80-100%) cytotoxicity was observed.
                    2
                      Neutralization control indicates the highest dilution of the endpoint titer where compound inhibited virus CPE in the wells after neutralization
                    3
                     Virus titers of the test sample or virus control (VC) in log10 CCID50 of virus per 0.1 ml
                    4
                      LRV (log reduction value) is the reduction of virus in the test sample compared to the virus control.




    96              Stoma Edu J. 2021;8(2): 95-99                                                                    pISSN 2360-2406; eISSN 2502-0285
Abdelahhad Barbour, et all
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temperature (22 ± 2°C) for 1 or 5 minutes as indicated    spread especially in high-risk disease transmission




                                                                                                                      Original Articles
in Tab. 1. The assay was neutralized by a 1/10            settings e.g., hospitals, long-term care facilities, and
dilution in MEM 2% FBS, 50 μg/mL gentamicin. For          vulnerable populations. One viable approach is to
quantification, the surviving virus from each sample      reduce viral loads in the oral and nasal cavities, which
was quantified by standard end-point dilution assay.      can be achieved by locally neutralizing viruses that
Briefly, the neutralized samples were pooled and          have entered these cavities with over-the-counter
serially diluted using eight log10 dilutions in a test    oral and/or nasal sprays with virucidal properties. In
medium. Then 100 μL of each dilution was plated           our current study, Flavobac based products exhibited
into quadruplicate wells of 96-well plates containing
                                                          excellent virucidal activities towards SARS-CoV-2
80-90% confluent Vero E6 cells (ATCC CRL-1586). The
                                                          when tested in vitro. These products can be used
toxicity controls were added to an additional 4 wells
                                                          as supplementary preventative measures to reduce
of Vero E6 cells and 2 of those wells at each dilution
were infected with the virus to serve as neutralization   exposure to infectious droplets, thus potentially
controls, ensuring that residual sample in the titer      reducing the person-to-person transmission risk in
assay plate did not inhibit growth and detection of       close contact situations. Nasal and oral antisepsis
the surviving virus. Plates were incubated at 37 ± 2°C    has been recommended as part of a comprehensive
with 5% CO2 for 5 days. Each well was then scored         plan to reduce the likelihood of virus transmission
for the presence or absence of an infectious virus.       by reducing the number of active aerosolized virus
The titers were determined using the Reed-Muench          particles from the nasal passages and oral cavity
(1948) equation [17] and the log reduction value          [9,18,19].
(LRV) of each compound compared to the negative           The American Dental Association and the Center for
(water) control was calculated.                           Disease Control and Prevention (CDC) guidelines
                                                          for minimizing the risk of COVID-19 transmission
3. RESULTS                                                advise the use of effective mouthwash before all
                                                          procedures [20]. Bioflavonoid-based products like
Flavobac BCL aqueous solution showed to have              Flavobac are known to be rich in plant polyphenols
potent antiviral activities by reducing SARS-CoV-2        which have been shown to have good antiviral
viral titer below the limit of detection (LoD) at all     (including SARS-CoV-2), antioxidant, antibacterial
concentrations tested in vitro. We have tested various
                                                          and anti-inflammatory properties [21]. A recent
concentrations to ensure that we identify the optimal
                                                          study has suggested that the anti-SARS-CoV-2
concentration of Flavobac BCL against SARS-COV-2.
                                                          activities of plant-derived natural polyphenols can
Flavobac BCL is a key ingredient of the formulation
OSI-20210203. The latter is the commercialized            be mediated by RNA dependent RNA polymerase
product (Cold & Flu Guard). Because of differences        (RdRp) inhibition which may represent an effective
in cytotoxicity, the lower concentrations had higher      therapy for SARS-CoV-2 infections [22]. In a sepa-
LRV values with LRV>2.9 at 2% and 1% and LRV>1.9          rated study, Jo et al found that many flavonoids
at 5% and 10%, respectively (Table 1). Furthermore,       were able to block the proteolytic activity of SARS-
Virus titers and LRV of SARS-CoV-2 after incubation       CoV-2 3CLpro, an essential enzyme controlling the
with Flavobac commercial solutions OSI-20210203A          virus replication life cycle [23]. Since Flavobac is a
and OSI-20210203B reduced the virus below the limit       mixture of plant-based bioflavonoids, it is believed
of detection (LRV>3.0). Each Flavobac containing          to exhibit similar modes of action towards SARS-
solution evaluated was effective at reducing >3 log10     CoV-2. Hence, scientists are recommending the use
CCID50 infectious virus, from 4.7 log10 CCID50/0.1 mL     of such products to reduce the spread of SARS-Cov-2
to <1.7 log10 CCID50/0.1 mL. A consistent reduction       [24] while we wait for a broad immunity conferred by
in virus titre was observed for SARS-CoV-2 viruses at     the new vaccines.
all concentrations of Flavobac solution tested and        The limitation of the current study is the lack of key
with a contact time of 1 or 5 minutes. The reductions     information on whether the tested product can
in virus titre were >1.9 log10 CCID50/mL for Flavobac     work in an actual in vivo environment and exhibit
5 and 10%, equating to >98.7% reduction; >2.9
                                                          the same virucidal activities when used by human
log10 CCID50/mL for Flavobac 1 and 2%, equating
                                                          consumers as a nasal spray. Further research is
to >99.8% reduction; and >3.0 Log10 CCID50/mL,
                                                          required by testing Flavobac in clinical trials to assess
equating to >99.9% reduction for OSI-202103, the
commercial formulation of Flavobac.                       its biological activities in preventing the spread
                                                          of the virus, As the world is now inching towards
4. DISCUSSION                                             gradually returning routine societal and economic
                                                          activities to pre-pandemic level, the heightened
In this era of emerging infectious diseases caused        fear of a post-pandemic outbreak looms as the virus
by respiratory tract viruses especially SARS-Cov-2,       still lurks and relatively little is known about the key
finding new alternative biomedical tools based            parameters that could shape the future course of the
on natural products is important to suppress viral        pandemic [25].


Stoma Edu J. 2021;8(2): 95-99                                            pISSN 2360-2406; eISSN 2502-0285                97
                    Efficacy of FLAVOBAC™ against SARS-CoV-2
www.stomaeduj.com



                    The challenge in nasal antisepsis is to find effective                   CONFLICT OF INTEREST
Original Articles   topical preparations which are safe to use. Oral and                     Dr. Glogauer is the Chief Scientific Officer for Oral Sciences. Oral
                    nasal solutions infused with Flavobac, a natural                         Sciences is the developer of this rinse product. The rest of the
                    bioflavonoid complex, with broad virucidal efficacy,                     authors declare no conflict of interest. Dr. Glogauer is the Chief
                    has demonstrated efficacy to kill 99.9% of SARS-                         Scientific Officer for Oral Sciences. Oral Sciences is the developer
                    CoV-2 and it may provide a safe and protective                           of this rinse product. The rest of the authors declare no conflict
                    solution for people within viruses-aerosolized places                    of interest.
                    like workplaces, gym, restaurant, schools or even for
                    people who are at a higher risk of respiratory viral                     ACKNOWLEDGMENTS
                    complications due to other health complications                          None.


                    5. CONCLUSION                                                            AUTHOR CONTRIBUTIONS
                                                                                             AB, MG contributed to the concept, design, and data analysis
                    Current public health recommendations emphasize                          of the study and wrote the manuscript. MM performed the
                    the need to break the person-to-person viral                             experiments. GD, HL contributed to the data analysis and edited
                    transmission primarily through social separation,                        the manuscript.
                    hand hygiene and surface disinfection. Flavobac
                    deactivated SARS-CoV-2 virus tested from 98.8%                           FUNDING
                    to > 99.9% when incubated with the virus for 1 to                        Oral Science International funded this study.
                    5 minutes at 22°C. The results indicate that Flavobac
                    oral and nasal spray could potentially be used to                        COMPETING INTERESTS
                    neutralize SARS-CoV-2 and reduce viral transmission.                     The authors declare that they have no competing interests.
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    98              Stoma Edu J. 2021;8(2):95-99                                                                pISSN 2360-2406; eISSN 2502-0285
Abdelahhad BARBOUR
                                                                                                                                       www.stomaeduj.com



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                                                                           Abdelahhad BARBOUR
                                                                             MSc, PhD, Postdoctoral Fellow
                                                                                       Faculty of Dentistry
                                                                                     University of Toronto
                                                                                     Toronto, ON, Canada


CV
Dr. Abdelahhad Barbour is a Postdoctoral scientist and research coordinator of the COVID-19 saliva testing project at the
Faculty of Dentistry, University of Toronto. The project aims to document rates of COVID-19 infection and immune responses to
vaccination among trainees, faculty, and staff in Canadian dental schools. Dr. Barbour obtained his PhD in Molecular Microbiology
from the University of Malaya, Malaysia with a thesis entitled “Characterisation and mechanism of action of lantibiotics produced
by Streptococcus salivarius”. He is an expert in the fields of antimicrobial peptides, microbial genomics, oral microbiome and
probiotics developments. Areas of interest in the research activity: Host-microbiome interactions, neutrophils-pathogens
signaling, COVID-19 saliva testing, antibiotic resistance, microbial genomics.



Questions
1. What are bioflavonoids?
qa. Synthetic substance;
qb. Natural products derived from animal origin;
qc. Natural products derived from fruits and vegetables;
qd. Antibiotics produced by soil microorganisms.

2. What are the biological activities of bioflavonoids?
qa. Antimicrobial;
qb. Antiviral;
qc. Antifungal;
qd. ll mentioned above.

3. What is the main composition of FLAVOBAC™?

qa. Soluble bioflavonoids and hydroxylated phenolic structures;
qb. Antimicrobial peptides;
qc. Polysaccharides;
qd. Lipids.

4. FLAVOBAC™ deactivated the SARS-CoV-2 virus at the following levels:
qa. 10-20%;
qb. Less than 50%;
qc. Less than 80%;
qd. More than 95%.



Stoma Edu J. 2021;8(2):95-99                                                        pISSN 2360-2406; eISSN 2502-0285                    99